2-((3-Trifluoromethyl)phenyl)histamine dimaleate | CAS 162049-83-4

Element: trifluoromethyl dimaleate histamine phenyl

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Identification

2-((3-Trifluoromethyl)phenyl)histamine dimaleate

CAS:

162049-83-4

EINECS:

Molecular Formula:

C₁₂H₁₂F₃N₃.2C₄H₄O₄

MDL:

SMILES:

C1=CC(=CC(=C1)C(F)(F)F)C2=NC=C(N2)CCN.C(=CC(=O)O)C(=O)O.C(=CC(=O)O)C(=O)O

Synonym:

2-((3-trifluoromethyl)phenyl)histamine d

Description

2-((3-Trifluoromethyl)phenyl)histamine dimaleate has been found to be the most potent and selective H₁ histamine receptor agonist of a panel of compounds in functional in vitro studies on histamine H₂, H₃, and other neurotransmitter receptors. It showed better potency at the guinea pig H₁ histamine receptor than at the human H₁ histamine receptor (pK_i = 5.9). The selectivity of 2-((3-Trifluoromethyl)phenyl)histamine dimaleate was found to be 2138 (H₁:H₂), > 64 (H₁:H₃), 1000 (H₁:M₃), 105 (H₁: α1), 708 (H₁:β1), and 71 (H₁:5HT_2A). This substance does not cross the blood-brain barrier.

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Data is processed

Properties for 2-((3-Trifluoromethyl)phenyl)histamine dimaleate

Molecular Weight:

487.38 g·mol−1

Melting point:

227° C

Solubility:

H₂O: ~20 mg/mL

Safety & Transport Information

Risk Codes:

R25 - Toxic if swallowed
R37/38 - Irritating to respiratory system and skin
R41 - Risk of serious damage to eyes

Safety Codes:

S26 - In case of contact with eyes, rinse immediately with plenty of water and seek medical advice
S39 - Wear eye/face protection
S45 - In case of accident or if you feel unwell seek medical advice immediately (show the label where possible)

Hazard Symbols:

Storage temperature :

2-8°C

RID/ADR certification :

UN 2811 6.1 / PG 3

Alternative Distributors of [2-((3-Trifluoromethyl)phenyl)histamine dimaleate]

Producers or manufacturers change the product range from time to time. Currently there are no other manufacturers known.

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